Photostability of Topoisomerase I Inhibitor Conjugated IgG1 Antibody-Drug Conjugates: Characterization Study and Degradation Mechanism Analysis
Bioconjug Chem. 2025 Nov 22. doi: 10.1021/acs.bioconjchem.5c00485. Online ahead of print. ABSTRACT DNA topoisomerase I (TOP1) inhibitor-based antibody-drug conjugates (ADCs) incorporating photosensitive camptothecin (CPT) analogs …